Protease Inhibitors and Phosphatase Inhibitors
MilliporeSigma™ Calbiochem™ Wiskostatin
A cell-permeable N-alkylated carbazole derivative that selectively blocks actin filament assembly.
MilliporeSigma™ Calbiochem™ 1400W
A selective, cell-permeable, irreversible, slow, tight-binding inhibitor of inducible nitric oxide synthase (iNOS; Kd = 7 nM).
MilliporeSigma™ Calbiochem™ NMD Inhibitor
A cell-permeable inhibitor of nonsense-mediated mRNA decay (NMD) that enhances the stability of premature termination codon mutated p53 mRNA in N417 and HDQP-1 cells.
MilliporeSigma™ Calbiochem™ AhR Antagonist II, SR1
The AhR Antagonist II, SR1 controls the biological activity of AhR. This small molecule/inhibitor is primarily used for Biochemicals applications.
MilliporeSigma™ Calbiochem™ Ghrelin Receptor Antagonist, JMV 2959
A 1, 2, 4-triazole derived compound that acts as a potent ghrelin receptor (GHS-R1a) antagonist (IC50 = 32nM in a binding assay, dissociation constant Kb =
MilliporeSigma™ Calbiochem™ Sodium Butyrate
A short chain fatty acid that has been shown to induce apoptosis in colon carcinoma cell lines by a p53-independent pathway.
MilliporeSigma™ Calbiochem™ PPARβ/δ Antagonist, GSK3787
The PPARβ/δAntagonist II, PT-S58, also referenced under CAS 188591-46-0, controls the biological activity of PPARβ/δ. This small molecule/inhibitor is primarily used for Biochemicals applications.
MilliporeSigma™ Calbiochem™ TCPOBOP
The most potent known member of the phenobarbital-like class of cytochrome P450 (CYP)-inducing agents.
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MilliporeSigma™ Calbiochem™ Trypsin Inhibitor, Soybean
The Trypsin Inhibitor, Soybean, also referenced under CAS 9035-81-8, controls the biological activity of Trypsin. This small molecule/inhibitor is primarily used for Protease Inhibitors applications.
MilliporeSigma™ Calbiochem™ Cathepsin K Substrate II, Fluorogenic
An internally quenched, highly cathepsin K-selective, fluorogenic peptide substrate that is efficiently cleaved by CatK (
MilliporeSigma™ Calbiochem™ Chymotrypsin Substrate II, Fluorogenic
Sensitive fluorogenic substrate for the quantitative determination of chymotrypsin activity.
MilliporeSigma™ Calbiochem™ GBR 12909 Dihydrochloride
A potent inhibitor of dopamine active transporter (DAT, Ki = 1 nM, IC50 = 40 and 51nM) with >100 fold selectivity over noradrenalin and 5-HT re-uptake trans
MilliporeSigma™ Calbiochem™ QX-314
A quaternary lidocaine derivative, permanently charged, and lipophobic.
MilliporeSigma™ Calbiochem™ α-(Methylamino)isobutyric Acid
A glutamine transport inhibitor selective for Na+-dependent amino acid transport system A.
MilliporeSigma™ Calbiochem™ Dynamin Inhibitor IV, Hydroxy-Dynasore
The Dynamin Inhibitor IV, Hydroxy-Dynasore controls the biological activity of Dynamin. This small molecule/inhibitor is primarily used for Cell Signaling applications.